SCHEMBL9027809

SCHEMBL9027809

CCn1cc(C(=O)NC2CC3CCCC(C2)N3C)c(=O)c2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 14/20 0.60
CNR1 P21554 2/20 0.57
CNR2 P34972 2/20 0.57
HTR3E A5X5Y0 5/20 0.56
HTR3B O95264 5/20 0.56
HTR3D Q70Z44 5/20 0.56
HTR3C Q8WXA8 5/20 0.56
SLC22A2 O15244 1/20 0.56
CHRNB2 P17787 1/20 0.56
CHRNA3 P32297 1/20 0.56
CHRNA4 P43681 1/20 0.56
KCNH2 Q12809 1/20 0.56
SLC47A1 Q96FL8 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9028063 0.96 HTR3A (0.61) HTR3ACNR1CNR2HTR3EHTR3B
SCHEMBL9029141 0.91 CNR2 (0.63) HTR3ACNR1CNR2HTR3EHTR3B
SCHEMBL9027144 0.89 HTR3A (0.66) HTR3ACNR1CNR2HTR3EHTR3B
SCHEMBL9028258 0.87 HTR3A (0.60) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9027450 0.87 HTR3A (0.67) HTR3ACNR1CNR2HTR3EHTR3B
SCHEMBL16378030 0.86 CNR1 (0.57) HTR3ACNR1CNR2HTR3EHTR3B
SCHEMBL22416052 0.86 CNR1 (0.57) HTR3ACNR1CNR2HTR3EHTR3B
SCHEMBL22416267 0.86 HTR3A (0.58) HTR3ACNR1CNR2HTR3EHTR3B
SCHEMBL16692891 0.86 HTR3A (0.58) HTR3ACNR1CNR2HTR3EHTR3B
SCHEMBL9027739 0.86 HTR3A (0.58) HTR3ACNR1CNR2HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0494978-B1 HETEROCYCLIC COMPOUNDS WYETH JOHN & BROTHER LTD (GB) 1996-02-28 EP disclosed
US-5362734-A Certain benzo-quinolizine compounds and derivatives thereof AMERICAN HOME PRODUCTS CORPORATION (US) 1994-11-08 US disclosed
US-5225419-A Antagonist 5-hydroxytryptamine for treatment of nausea or vomiting JOHN WYETH & BROTHER, LIMITED (GB) 1993-07-06 US disclosed
US-5096901-A PHARMACOLOGICALLY ACTIVE AMIDES AND ESTERS CONTAINING AN AZABICYCLOALKANE MOIETY JOHN WYETH & BROTHER LIMITED (GB) 1992-03-17 US disclosed