SCHEMBL9028004

SCHEMBL9028004

CC(C)Oc1cccc(CC(=O)C2CC(CCN3CCN(C4CCCCC4)CC3)(c3cccc(Cl)c3)CCCN2)c1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.43
TACR2 P21452 1/20 0.43
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
DPP9 Q86TI2 1/20 0.38
HRH1 P35367 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9028158 0.95 TACR1 (0.44) TACR1TACR2DPP4DPP8DPP9
SCHEMBL9027626 0.92 TACR1 (0.51) TACR1TACR2
SCHEMBL9027873 0.91 TACR1 (0.41) TACR1TACR2HRH1HRH3
SCHEMBL9028446 0.90 TACR1 (0.42) TACR1TACR2HRH1
SCHEMBL9027525 0.90 TACR1 (0.43) TACR1TACR2HRH1KDM4EALDH1A1
SCHEMBL9026973 0.90 TACR1 (0.41) TACR1TACR2HRH1
SCHEMBL9027964 0.89 TACR1 (0.40) TACR1TACR2HRH1
SCHEMBL9027398 0.89 TACR1 (0.47) TACR1TACR2HRH1ALDH1A1
SCHEMBL9028989 0.88 TACR1 (0.43) TACR1TACR2HRH1
SCHEMBL9028402 0.88 TACR1 (0.40) TACR1TACR2HRH1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563133-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-10-08 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed