SCHEMBL9028402

SCHEMBL9028402

CC(C)Oc1cccc(CC(=O)C2CC(CCN3CCN(C4CCCCC4)CC3)(c3ccc(C(F)(F)F)c(C(F)(F)F)c3)CCCN2)c1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.40
TACR2 P21452 1/20 0.39
HRH1 P35367 1/20 0.38
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
BRS3 P32247 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9027834 0.95 TACR1 (0.39) TACR1TACR2HRH1BRS3KDM4E
SCHEMBL9027964 0.93 TACR1 (0.40) TACR1TACR2HRH1
SCHEMBL9027873 0.90 TACR1 (0.41) TACR1TACR2HRH1
SCHEMBL9028446 0.89 TACR1 (0.42) TACR1TACR2HRH1
SCHEMBL9027525 0.89 TACR1 (0.43) TACR1TACR2HRH1KDM4EALDH1A1
SCHEMBL9026973 0.89 TACR1 (0.41) TACR1TACR2HRH1
SCHEMBL9027626 0.89 TACR1 (0.51) TACR1TACR2
SCHEMBL9027398 0.88 TACR1 (0.47) TACR1TACR2HRH1ALDH1A1
SCHEMBL9028004 0.88 TACR1 (0.43) TACR1TACR2HRH1KDM4EALDH1A1
SCHEMBL9028989 0.87 TACR1 (0.43) TACR1TACR2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563133-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-10-08 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed