SCHEMBL9028776

SCHEMBL9028776

COC(=O)c1ccc(CC(=O)c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.52
CA1 P00915 3/20 0.52
CA2 P00918 3/20 0.52
CA9 Q16790 3/20 0.52
CA14 Q9ULX7 3/20 0.52
LOXL2 Q9Y4K0 1/20 0.50
NPC1 O15118 2/20 0.49
MAPT P10636 2/20 0.49
RAB9A P51151 2/20 0.49
PTGS2 P35354 1/20 0.49
GSR P00390 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
FBP1 P09467 1/20 0.47
CYP4A11 Q02928 2/20 0.46
POLB P06746 2/20 0.46
MAPK1 P28482 1/20 0.46
HPGD P15428 1/20 0.45
CYP4F2 P78329 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7625358 1.00 CA12 (0.52) CA12CA1CA2CA9CA14
SCHEMBL2228992 0.85 CA1 (0.62) CA12CA1CA2CA9CA14
SCHEMBL7619212 0.83 SRD5A2 (0.56) CA12CA1CA2CA9CA14
SCHEMBL6180942 0.83 NPC1 (0.63) NPC1RAB9APTGS2GSRKMT2A
SCHEMBL6970870 0.81 PTGS2 (0.53) PTGS2GSRKMT2A
SCHEMBL4772305 0.81 PTGS2 (0.53) PTGS2GSRKMT2A
SCHEMBL6341279 0.81 PTGS2 (0.51) MAPTPTGS2GSR
SCHEMBL8602859 0.81 MAPT (0.59) MAPTPTGS2GSR
SCHEMBL14156906 0.81 CA1 (0.69) CA12CA1CA2CA9CA14
SCHEMBL7165400 0.81 TSHR (0.66) CA1CA2LOXL2NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739340-A1 PHENYL HETEROCYCLES AS COX-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1996-10-30 EP disclosed