SCHEMBL9028853

SCHEMBL9028853

COc1ccc(CNC(=O)C(C)Cl)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.68
MEN1 O00255 2/20 0.66
KMT2A Q03164 2/20 0.66
MAPK1 P28482 1/20 0.59
POLB P06746 1/20 0.57
ATM Q13315 1/20 0.56
EPHX2 P34913 1/20 0.54
CTSD P07339 3/20 0.54
TDP1 Q9NUW8 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
LMNA P02545 1/20 0.53
GAA P10253 2/20 0.53
KDM4E B2RXH2 1/20 0.53
CYP3A4 P08684 1/20 0.53
ALOX15 P16050 1/20 0.53
TSHR P16473 1/20 0.53
RAB9A P51151 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9781286 0.90 ALDH1A1 (0.69) ALDH1A1MEN1KMT2AMAPK1POLB
SCHEMBL5018017 0.84 ALDH1A1 (0.66) ALDH1A1MEN1KMT2AMAPK1POLB
SCHEMBL13074346 0.81 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AMAPK1POLB
SCHEMBL6093048 0.81 ERCC1 (0.66) ALDH1A1MEN1KMT2AMAPK1POLB
SCHEMBL18814446 0.80 ALDH1A1 (0.59) ALDH1A1MEN1KMT2AEPHX2SMN1; SMN2
SCHEMBL6171639 0.80 ALDH1A1 (0.78) ALDH1A1MEN1KMT2AMAPK1POLB
SCHEMBL2936661 0.80 ALDH1A1 (0.78) ALDH1A1MEN1KMT2AMAPK1POLB
SCHEMBL2846636 0.80 ALDH1A1 (0.78) ALDH1A1MEN1KMT2AMAPK1POLB
SCHEMBL28721168 0.79 ALDH1A1 (0.68) ALDH1A1MEN1KMT2AMAPK1POLB
SCHEMBL20456221 0.79 ALDH1A1 (0.71) ALDH1A1MEN1KMT2APOLBATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700389-A1 ANTI-ARRHYTHMIC N-SUBSTITUTED 3-BENZAZEPINES OR ISOQUINOLINES SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1996-03-13 EP disclosed
WO-1994027971-A1 ANTI-ARRHYTHMIC N-SUBSTITUTED 3-BENZAZEPINES OR ISOQUINOLINES SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1994-12-08 WO disclosed