SCHEMBL903018

SCHEMBL903018

Bc1cc(C(=O)O)cnc1OCC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.50
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
TSHR P16473 1/20 0.41
HCAR3 P49019 1/20 0.38
PLA2G4B P0C869 1/20 0.38
P4HTM Q9NXG6 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 2/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27371818 0.81 TSHR (0.53) MAPTCYP2C9CYP2C19TSHRP4HTM
SCHEMBL6233391 0.81 MAPT (0.51) MAPTCYP2C9CYP2C19TSHRHCAR3
SCHEMBL17069361 0.80 MAPT (0.50) MAPTCYP2C9CYP2C19KMT2APOLB
SCHEMBL3369108 0.80 MAPT (0.50) MAPTCYP2C9CYP2C19TSHRHCAR3
SCHEMBL899216 0.80 MAPT (0.50) MAPTCYP2C9CYP2C19TSHRP4HTM
SCHEMBL12582009 0.79 KMT2A (0.42) HCAR3RXRARXRBKMT2AALOX15
SCHEMBL2121557 0.76 ALDH1A1 (0.47) MAPTCYP2C9CYP2C19POLBALOX15
SCHEMBL12845747 0.73 HCAR2 (0.47) CYP2C9CYP2C19HCAR3P4HTMKMT2A
SCHEMBL6359091 0.72 KMT2A (0.48) MAPTCYP2C9CYP2C19TSHRKMT2A
SCHEMBL8881108 0.71 TSHR (0.53) MAPTCYP2C9CYP2C19TSHRP4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012042433-A1 N1-PYRAZOLOSPIROKETONE ACETYL-CoA CARBOXYLASE INHIBITORS PFIZER INC. (US) 2012-04-05 WO disclosed