SCHEMBL9030749

SCHEMBL9030749

O=C1CCCN1CC#CCc1ncc[nH]1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.52
CHRM5 P08912 4/20 0.52
CHRM1 P11229 4/20 0.52
CHRM3 P20309 3/20 0.50
CYP2D6 P10635 2/20 0.50
CYP1A2 P05177 1/20 0.50
CHRM4 P08173 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
ALDH1A1 P00352 2/20 0.47
LMNA P02545 2/20 0.47
APEX1 P27695 2/20 0.47
PMP22 Q01453 2/20 0.47
TSHR P16473 1/20 0.47
ALOX12 P18054 1/20 0.47
NFKB1 P19838 1/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12471192 0.80 ALOX15 (0.54) CHRM2CHRM5CHRM1CYP1A2CYP2C9
SCHEMBL9029943 0.71 CHRM2 (0.71) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL6930591 0.70 ALOX15 (0.46) ALDH1A1
SCHEMBL9646306 0.69 CHRM2 (0.51) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL9029818 0.69 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL9029969 0.69 CHRM2 (0.56) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL31263727 0.68 CHRM2 (0.93) CHRM2CHRM5CHRM1CHRM3CYP2D6
Oxotremorine SCHEMBL2128 0.68 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL9029739 0.68 CHRM2 (0.68) CHRM2CHRM5CHRM1CHRM3CYP2D6
SCHEMBL9029648 0.68 CHRM2 (0.56) CHRM2CHRM5CHRM1CHRM3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426714-B1 ACETYLENIC IMIDAZOLES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY UPJOHN CO (US) 1996-04-03 EP claimed