SCHEMBL9030764

SCHEMBL9030764

CCCCS(=O)(=O)CCc1ccc(C(=N)N)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 3/20 0.45
ST14 Q9Y5Y6 1/20 0.44
F2 P00734 4/20 0.44
PRSS1 P07477 2/20 0.44
PRSS2 P07478 2/20 0.44
PRSS3 P35030 2/20 0.44
PLG P00747 1/20 0.44
C1S P09871 1/20 0.44
F10 P00742 3/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
CA2 P00918 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SPHK2 Q9NRA0 2/20 0.41
SPHK1 Q9NYA1 2/20 0.41
ITGB3 P05106 3/20 0.41
ITGA2B P08514 3/20 0.41
RARB P10826 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555919 0.86 MRGPRX1 (0.46) MRGPRX1ST14F2PRSS1PRSS2
SCHEMBL8995527 0.80 PRSS1 (0.55) ST14PRSS1PRSS2PRSS3F10
Hydrochloric Acid SCHEMBL5884387 0.79 PRSS1 (0.53) ST14F2PRSS1PRSS2PRSS3
SCHEMBL9649899 0.79 ESR1 (0.55) PRSS1PRSS2PRSS3F10LOXL2
SCHEMBL9650566 0.77 ESR1 (0.58) SPHK2SPHK1RARB
SCHEMBL9647294 0.77 ESR1 (0.58) SPHK2SPHK1RARB
SCHEMBL9650482 0.77 ESR1 (0.58) SPHK2SPHK1RARB
SCHEMBL9650690 0.77 ESR1 (0.58) SPHK2SPHK1RARB
Hydrochloric Acid SCHEMBL7798271 0.77 SPHK1 (0.56) PRSS1PRSS2PRSS3F10LOXL2
SCHEMBL9650583 0.77 ESR1 (0.58) SPHK2SPHK1RARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed