SCHEMBL8555919

SCHEMBL8555919

CCCCS(=O)(=O)Cc1ccc(C(=N)N)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 3/20 0.46
PRSS1 P07477 5/20 0.44
PRSS2 P07478 5/20 0.44
PRSS3 P35030 5/20 0.44
F10 P00742 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
F2 P00734 3/20 0.41
PLG P00747 1/20 0.41
C1S P09871 1/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
POLB P06746 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
ALOX15 P16050 1/20 0.40
BRCA1 P38398 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9030764 0.86 MRGPRX1 (0.45) MRGPRX1PRSS1PRSS2PRSS3F10
SCHEMBL8409513 0.79 KMT2A (0.48) PRSS1PRSS2PRSS3F10LOXL2
SCHEMBL9030595 0.78 MRGPRX1 (0.46) MRGPRX1PRSS1PRSS2PRSS3F10
SCHEMBL9030747 0.78 PRSS1 (0.55) MRGPRX1PRSS1PRSS2PRSS3F10
SCHEMBL9030039 0.78 THRA (0.49) MRGPRX1PRSS1PRSS2PRSS3F2
Hydrochloric Acid SCHEMBL8410206 0.76 CYP2C19 (0.39) PRSS1PRSS2PRSS3F10F2
SCHEMBL16489292 0.76 PRSS1 (0.46) PRSS1PRSS2PRSS3F10LOXL2
SCHEMBL9030515 0.76 MRGPRX1 (0.47) MRGPRX1PRSS1PRSS2PRSS3F2
SCHEMBL6652748 0.75 KMT2A (0.41) ALDH1A1LMNAPOLBRAB9ASMN1; SMN2
SCHEMBL8995527 0.74 PRSS1 (0.55) PRSS1PRSS2PRSS3F10LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832076-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-04-01 EP disclosed
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed