SCHEMBL9030784

SCHEMBL9030784

CCCC1CC=C(c2ccc(-c3ccc(Cl)c(F)c3)nc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 3/20 0.39
TYRO3 Q06418 3/20 0.39
MERTK Q12866 3/20 0.39
GAS6 Q14393 3/20 0.39
CYP11B1 P15538 4/20 0.35
CYP11B2 P19099 4/20 0.35
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ESR2 Q92731 1/20 0.34
GRM2 Q14416 2/20 0.33
KMO O15229 2/20 0.33
CCNT1 O60563 1/20 0.32
CDK9 P50750 1/20 0.32
GRIN2B Q13224 1/20 0.32
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10015003 0.88 ESR2 (0.40) CYP11B1CYP11B2NPC1RAB9AESR2
SCHEMBL12254194 0.83 ESR2 (0.33) FLT3TYRO3MERTKGAS6ESR2
SCHEMBL10015005 0.80 ESR2 (0.42) FLT3TYRO3MERTKGAS6NPC1
SCHEMBL12254134 0.79 FLT3 (0.34) FLT3TYRO3MERTKGAS6
SCHEMBL10015006 0.77 FLT3 (0.33) FLT3TYRO3MERTKGAS6
SCHEMBL9029730 0.77 CYP2C9 (0.38) CYP11B1CYP11B2NPC1TP53PKM
SCHEMBL9029726 0.77 CYP2C9 (0.38) CYP11B1CYP11B2NPC1TP53PKM
SCHEMBL9019416 0.76 ESR2 (0.43) CYP11B1CYP11B2NPC1RAB9AESR2
SCHEMBL10015008 0.76 FLT3 (0.33) FLT3TYRO3MERTKGAS6
SCHEMBL11190434 0.74 ESR2 (0.54) FLT3TYRO3MERTKGAS6NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456793-B1 HALOPHENYL SUBSTITUTED HETEROCYCLIC DERIVATIVES MERCK PATENT GMBH (DE) 1996-10-23 EP disclosed
WO-1991009016-A2 HALOPHENYL SUBSTITUTED HETEROCYCLIC DERIVATIVES MERCK PATENT GMBH (DE) 1991-06-27 WO disclosed
WO-1991009016-A1 HALOPHENYL SUBSTITUTED HETEROCYCLIC DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-06-27 WO disclosed