SCHEMBL9032151

SCHEMBL9032151

CCCn1c(=O)n2c(C)nnc2c2[nH]cnc21

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 19/20 0.65
PDE4B Q07343 19/20 0.65
PDE4C Q08493 19/20 0.65
PDE4D Q08499 19/20 0.65
ADORA2A P29274 12/20 0.65
ADORA2B P29275 10/20 0.65
ADORA3 P0DMS8 1/20 0.55
HPGD P15428 1/20 0.55
ADORA1 P30542 1/20 0.55
BLM P54132 1/20 0.55
PDE3A Q14432 1/20 0.55
HSD17B10 Q99714 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9032044 0.82 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9029804 0.81 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9031869 0.80 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL515771 0.79 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9030884 0.79 PNP (0.57) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL9031532 0.79 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DADORA2A
Ammonia Solution, Strong SCHEMBL10420651 0.78 PDE4A (0.97) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9029959 0.78 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL4623455 0.77 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9765669 0.77 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP disclosed
US-5173492-A Bronchodilator agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-12-22 US disclosed
EP-0417790-A2 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-20 EP disclosed