SCHEMBL9032893

SCHEMBL9032893

COCN1C(C)=C(C(=O)O)C(c2cccc([N+](=O)[O-])c2)C(C(=O)O)=C1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.57
CYP3A4 P08684 5/20 0.57
CYP2C9 P11712 5/20 0.57
CYP2C19 P33261 5/20 0.57
MAPT P10636 3/20 0.57
CYP2D6 P10635 3/20 0.57
TSHR P16473 3/20 0.57
NFKB1 P19838 3/20 0.57
LMNA P02545 3/20 0.57
GMNN O75496 1/20 0.57
BLM P54132 1/20 0.57
PMP22 Q01453 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
PDE1C Q14123 1/20 0.56
CACNA1F O60840 8/20 0.56
CACNA1D Q01668 8/20 0.56
CACNA1S Q13698 8/20 0.56
CACNA1C Q13936 8/20 0.56
ADORA3 P0DMS8 1/20 0.56
HIF1A Q16665 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9033536 1.00 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL9033652 0.95 MAPT (0.65) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL9032956 0.95 MAPT (0.65) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL9032974 0.95 MAPT (0.65) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL9033294 0.95 MAPT (0.65) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL9032948 0.90 CYP1A2 (0.70) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL20801670 0.89 CYP1A2 (0.55) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL7286552 0.89 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL7286542 0.89 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL9031678 0.88 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C9CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0474129-B1 1,4-Dihydropyridine derivatives and process for preparing the same ACHIWA KAZUO (JP) 1996-12-18 EP disclosed
US-5336774-A 1,4-dihydropyridine 3,5 carboxyl compounds ACHIWA KAZUO (JP) 1994-08-09 US disclosed
US-5234821-A Process for preparing 1,4 dihydropyridine compounds ACHIWA KAZUO (JP) 1993-08-10 US disclosed
EP-0474129-A2 1,4-Dihydropyridine derivatives and process for preparing the same Achiwa, Kazuo (JP) 1992-03-11 EP disclosed