SCHEMBL9034706

SCHEMBL9034706

COc1cc2ccc(C(=O)O)cc2nc1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA4 P22748 2/20 0.53
CA6 P23280 2/20 0.53
CA7 P43166 2/20 0.53
CA9 Q16790 2/20 0.53
CA14 Q9ULX7 2/20 0.53
TPMT P51580 1/20 0.53
RAB9A P51151 3/20 0.53
HTT P42858 2/20 0.53
LMNA P02545 2/20 0.53
MAPK1 P28482 1/20 0.53
KDM4E B2RXH2 1/20 0.50
PDGFRB P09619 1/20 0.48
PDGFRA P16234 1/20 0.48
TSHR P16473 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
RARA P10276 1/20 0.45
RARB P10826 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9036638 0.98 CA12 (0.51) CA12CA1CA2CA4CA6
SCHEMBL8156878 0.88 ALDH1A1 (0.43) HTTLMNAMAPK1TSHRHSD17B10
SCHEMBL4946900 0.76 KDM4E (0.70) CA12CA1CA2CA4CA6
SCHEMBL2671576 0.76 KDM4E (0.54) CA12CA1CA2CA4CA6
SCHEMBL22672508 0.75 TDP1 (0.54) CA12CA1CA2CA4CA6
SCHEMBL13230262 0.73 BACE1 (0.43) RAB9AHTTKDM4EPDGFRBPDGFRA
SCHEMBL360580 0.73 KDM4E (0.60) CA12CA1CA2CA4CA6
SCHEMBL9319496 0.72 KDM4E (0.57) CA12CA1CA2CA4CA6
SCHEMBL8155683 0.72 UGT2B7 (0.42) HTTLMNAPDGFRBPDGFRATSHR
SCHEMBL8148257 0.72 CYP2A6 (0.44) RAB9AHTTLMNAMAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103601674-B A kind of suppress dipeptides kininase compound and preparation method and purposes ZHEJIANG UNIVERSITY (CN) 2015-09-23 CN disclosed
CN-1350524-A Quinoline derivatives as inhibitors of MEK enzymes ASTRAZENECA AB (SE) 2002-05-22 CN disclosed
CN-1195988-A Immunosuppressant TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-10-14 CN disclosed
CN-1181376-A Production of benzophenone derivatives TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-05-13 CN disclosed
CN-1156453-A Process for preparing quinazoline or quinoline derivatives and intermediates therefor TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-08-06 CN disclosed
EP-0749426-A1 QUINOLINE OR QUINAZOLINE DERIVATIVES AS ANTI-INFLAMMATORY AGENTS, IN PARTICULAR FOR TREATING ARTHRITIS Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed
WO-1995024394-A1 QUINOLINE OR QUINAZOLINE DERIVATIVES AS ANTI-INFLAMMATORY AGENTS, IN PARTICULAR FOR TREATING ARTHRITIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-09-14 WO disclosed