SCHEMBL903681

SCHEMBL903681

Clc1ccc2c(c1)OCn1c-2c(Br)c2cc(Cl)ccc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.34
PIK3CB P42338 3/20 0.34
PIK3CG P48736 3/20 0.34
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10217252 0.81 PIK3CA (0.38) PIK3CAPIK3CBPIK3CGMAPTKDM4E
SCHEMBL10215147 0.70 HTR2A (0.39) PIK3CAPIK3CBPIK3CGHTR2AHTR2C
SCHEMBL10173672 0.69 MAPT (0.36) PIK3CAPIK3CBPIK3CGMAPTMEN1
SCHEMBL17613183 0.65 PIK3CA (0.39) PIK3CAPIK3CBPIK3CGMAPTMEN1
SCHEMBL10173675 0.64 PIK3CA (0.38) PIK3CAPIK3CBPIK3CGMAPTKDM4E
SCHEMBL9169246 0.60 MAOB (0.38) HTR2AHTR2CMAP3K14
SCHEMBL8980735 0.59 DPP4 (0.39) KDM4EMAP3K14
SCHEMBL14764759 0.59 PIK3CA (0.37) PIK3CAPIK3CBPIK3CGPIK3CD
SCHEMBL14765030 0.57 PIK3CA (0.61) PIK3CAPIK3CBPIK3CGKDM4EMEN1
SCHEMBL6862405 0.57 CA1 (0.36) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041014-A1 TETRACYCLIC INDOLE DERIVATIVES FOR TREATING HEPATITIS C VIRUS INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed