SCHEMBL6862405

SCHEMBL6862405

Nc1c2n(c3cc(Cl)ccc13)COC2=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
NTRK1 P04629 1/20 0.35
MAT2A P31153 4/20 0.34
IDO1 P14902 4/20 0.33
KMT2A Q03164 1/20 0.33
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32
NOS2 P35228 2/20 0.32
CA12 O43570 1/20 0.32
CA3 P07451 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA13 Q8N1Q1 1/20 0.32
CA14 Q9ULX7 1/20 0.32
CA5B Q9Y2D0 1/20 0.32
MAPK8 P45983 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31223911 0.62 MAT2A (0.46) NTRK1MAT2A
SCHEMBL903681 0.57 PIK3CA (0.34) KMT2A
SCHEMBL28277831 0.57 OPRK1 (0.42) MAT2AKMT2A
SCHEMBL25412172 0.57 MAT2A (0.41) MAT2AKMT2ANOS3NOS1NOS2
SCHEMBL25411473 0.57 MAT2A (0.41) MAT2ANOS3NOS1NOS2MAPK8
SCHEMBL30727441 0.56 MAT2A (0.50) NTRK1MAT2A
SCHEMBL22093343 0.56 MAT2A (0.72) MAT2A
SCHEMBL25410818 0.55 MAPK8 (0.38) NTRK1MAT2AKMT2ACA12CA9
SCHEMBL21979009 0.55 NQO2 (0.61) NTRK1MAT2A
SCHEMBL30901294 0.55 NQO2 (0.61) NTRK1MAT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011106650-A2 NOVEL P53-MDM2/P53-MDM4 ANTAGONISTS TO TREAT PROLIFERATIVE DISEASE UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2011-09-01 WO disclosed