SCHEMBL9037754

SCHEMBL9037754

NC(=Nc1ccc(CCNCc2cccc(Cl)c2)cc1)c1sccc1Cl

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 4/20 0.72
NOS1 P29475 3/20 0.72
NOS2 P35228 3/20 0.72
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
HDAC1 Q13547 1/20 0.44
CHRM2 P08172 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6953744 0.99 NOS3 (0.73) NOS3NOS1NOS2CYP1A2CYP3A4
SCHEMBL122446 0.84 NOS3 (1.00) NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL30007714 0.83 NOS3 (1.00) NOS3NOS1NOS2
SCHEMBL9037985 0.81 NOS3 (0.69) NOS3NOS1NOS2CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL6956568 0.80 NOS3 (0.70) NOS3NOS1NOS2CYP1A2CYP3A4
SCHEMBL9037749 0.79 CYP1A2 (0.51) NOS3NOS1NOS2CYP1A2CYP3A4
SCHEMBL6967979 0.78 NOS3 (0.88) NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL6953741 0.78 CYP1A2 (0.53) NOS3NOS1NOS2CYP1A2CYP3A4
SCHEMBL6967594 0.75 NOS3 (0.84) NOS3NOS1NOS2
SCHEMBL6962890 0.75 NOS3 (0.80) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1071746-C Amidine derivatives with nitric oxide synthetase activities ASTERA CO (SE) 2001-09-26 CN claimed
CN-1132505-A Amidine derivatives with nitric oxide synthetase activities ASTERA CO (SE) 1996-10-02 CN claimed
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP claimed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO claimed