SCHEMBL9037798

SCHEMBL9037798

CC(CCCc1cc(O)c(C(c2ccccc2)C2CC2)c(=O)o1)Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ELANE P08246 3/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
CYP2C9 P11712 5/20 0.32
VKORC1 Q9BQB6 2/20 0.32
MAPT P10636 1/20 0.32
LMNA P02545 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9201359 0.88 CYP2C9 (0.33) HTR2BSMN1; SMN2CYP2C9VKORC1LMNA
SCHEMBL6174391 0.87 HTR2B (0.46) HTR2BNPC1RAB9ASMN1; SMN2MTNR1A
SCHEMBL6173304 0.87 HTR2B (0.43) HTR2BNPC1RAB9ASMN1; SMN2ELANE
SCHEMBL6174697 0.85 HTR2B (0.43) HTR2BNPC1RAB9ASMN1; SMN2CYP2C9
SCHEMBL9194038 0.85 CYP2C9 (0.38) ELANECYP2C9VKORC1MAPT
SCHEMBL9199339 0.84 ELANE (0.47) NPC1RAB9ASMN1; SMN2ELANEMAPT
SCHEMBL9201135 0.84 ELANE (0.47) NPC1RAB9ASMN1; SMN2ELANEMAPT
SCHEMBL9199422 0.84 CYP2C9 (0.35) ELANECYP2C9VKORC1MAPT
SCHEMBL6174860 0.83 ELANE (0.33) HTR2BELANECYP2C9VKORC1MAPT
SCHEMBL6175617 0.83 ELANE (0.33) HTR2BRAB9AELANECYP2C9VKORC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed