SCHEMBL9038754

SCHEMBL9038754

CC(C)(C)OC(=O)CC[C@H](NC(=O)c1ccc(CCCc2c(N)nc(N)nc2Cl)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.47
GART P22102 1/20 0.45
ATIC P31939 1/20 0.45
TYMS P04818 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9217360 0.88 DHFR (0.35) DHFRGARTATIC
SCHEMBL9037720 0.86 DHFR (0.54) DHFRGARTATICTYMS
SCHEMBL9037088 0.85 DHFR (0.66) DHFR
SCHEMBL9037916 0.81 DHFR (0.69) DHFRGARTATICTYMS
SCHEMBL9088792 0.78 P2RY12 (0.43)
SCHEMBL9088784 0.78 P2RY12 (0.43)
SCHEMBL9343679 0.78 DHFR (0.54) DHFRGARTATICTYMS
SCHEMBL9343678 0.78 DHFR (0.54) DHFRGARTATICTYMS
SCHEMBL9556410 0.78 P2RY12 (0.42)
SCHEMBL9087240 0.78 P2RY12 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722440-A1 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1996-07-24 EP disclosed
EP-0722440-A4 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES LILLY CO ELI (US) 1996-06-04 EP disclosed
US-5426110-A Inhibiting dihydrofolate reductase in mammals and treating susceptible reoplasms ELI LILLY AND COMPANY (US) 1995-06-20 US disclosed
WO-1995009845-A1 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1995-04-13 WO disclosed