SCHEMBL9039550

SCHEMBL9039550

CCCCn1cccc1C(=O)NCCC(=O)OCC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.47
MAPT P10636 1/20 0.45
TNF P01375 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
ALDH1A1 P00352 2/20 0.40
CNR1 P21554 1/20 0.40
NAMPT P43490 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C19 P33261 2/20 0.39
POLB P06746 2/20 0.38
THRB P10828 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9041396 0.93 CNR2 (0.44) CNR2MAPTTNFSMN1; SMN2ALDH1A1
SCHEMBL9039339 0.87 CNR2 (0.43) CNR2MAPTTNFSMN1; SMN2ALDH1A1
SCHEMBL9037774 0.85 NPSR1 (0.47) CNR2SMN1; SMN2ALDH1A1CNR1NPC1
SCHEMBL6990088 0.83 NPC1 (0.57) MAPTALDH1A1NPC1RAB9AKDM4E
SCHEMBL6988747 0.82 CNR2 (0.55) CNR2MAPTCNR1NPC1RAB9A
SCHEMBL9039943 0.78 CYP3A4 (0.40) CNR2MAPTSMN1; SMN2ALDH1A1NAMPT
SCHEMBL23852583 0.77 TNF (0.54) CNR2TNFCNR1
SCHEMBL9037906 0.77 NPC1 (0.48) CNR2MAPTALDH1A1NPC1RAB9A
SCHEMBL23852674 0.76 TNF (0.50) CNR2TNFALDH1A1CNR1
SCHEMBL6991219 0.75 HRH4 (0.47) CNR2SMN1; SMN2ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441349-B1 Pyrroloazepine derivatives SUNTORY LTD (JP) 1996-01-03 EP disclosed
US-5416082-A Antiserotonine agents SUNTORY LIMITED (JP) 1995-05-16 US disclosed
US-5391731-A Useful therapeutics for circulatory diseases SUNTORY LIMITED (JP) 1995-02-21 US disclosed
US-5206239-A Cardiovascular disorders SUNTORY LIMITED (JP) 1993-04-27 US disclosed