SCHEMBL9037774

SCHEMBL9037774

CCCCn1cccc1C(=O)NCCC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
CNR2 P34972 2/20 0.43
CNR1 P21554 1/20 0.43
NAAA Q02083 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
LMNA P02545 1/20 0.40
ALDH1A1 P00352 2/20 0.40
S1PR1 P21453 2/20 0.40
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
GCGR P47871 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PLA2G2A P14555 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037906 0.92 NPC1 (0.48) NPSR1NPC1RAB9ACNR2NAAA
SCHEMBL6993812 0.86 NPC1 (0.47) NPSR1NPC1RAB9ACNR2LMNA
SCHEMBL9039550 0.85 CNR2 (0.47) NPC1RAB9ACNR2CNR1TSHR
SCHEMBL6988127 0.80 RAB9A (0.68) NPC1RAB9ASMN1; SMN2
SCHEMBL6992210 0.78 CNR2 (0.64) NPC1RAB9ACNR2CNR1KDM4E
SCHEMBL1606849 0.78 CNR2 (0.42) NPSR1CNR2CNR1LMNAALDH1A1
SCHEMBL9041396 0.76 CNR2 (0.44) NPC1RAB9ACNR2ALDH1A1SMN1; SMN2
SCHEMBL5252375 0.75 CNR2 (0.43) NPSR1CNR2CNR1LMNAALDH1A1
SCHEMBL9852009 0.74 BRD4 (0.44) NPC1RAB9ACNR2CNR1LMNA
SCHEMBL5657254 0.74 NPC1 (0.64) NPC1RAB9ANAAATSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441349-B1 Pyrroloazepine derivatives SUNTORY LTD (JP) 1996-01-03 EP disclosed
US-5416082-A Antiserotonine agents SUNTORY LIMITED (JP) 1995-05-16 US disclosed
US-5391731-A Useful therapeutics for circulatory diseases SUNTORY LIMITED (JP) 1995-02-21 US disclosed
US-5206239-A Cardiovascular disorders SUNTORY LIMITED (JP) 1993-04-27 US disclosed
EP-0441349-A1 Pyrroloazepine derivatives SUNTORY LIMITED (JP) 1991-08-14 EP disclosed