SCHEMBL9039873

SCHEMBL9039873

CS(=O)(=O)Nc1ccc2c(c1)CC(C1CCc3cc(C#N)ccc3C1)C1(CCNCC1)O2

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.50
DRD2 P14416 2/20 0.36
DRD3 P35462 2/20 0.36
BRD4 O60885 1/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR6 P50406 1/20 0.34
PGR P06401 2/20 0.34
MCHR1 Q99705 1/20 0.32
KDM1A O60341 1/20 0.32
ALDH2 P05091 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9041198 0.84 KCNH2 (0.37) KCNH2
SCHEMBL7388072 0.84 KCNH2 (0.48) KCNH2DRD2DRD3BRD4HTR2A
SCHEMBL7383232 0.84 KCNH2 (0.53) KCNH2DRD2DRD3BRD4HTR2A
Hydrochloric Acid SCHEMBL7359212 0.84 KCNH2 (0.48) KCNH2DRD2DRD3BRD4PGR
SCHEMBL7389329 0.79 KCNH2 (0.50) KCNH2DRD2DRD3KDM1A
SCHEMBL7384445 0.77 KCNH2 (0.48) KCNH2DRD2DRD3
Hydrochloric Acid SCHEMBL8832236 0.75 KCNH2 (0.46) KCNH2DRD2DRD3
SCHEMBL8563993 0.73 KCNH2 (0.77) KCNH2DRD2HTR2A
SCHEMBL8831674 0.73 KCNH2 (0.77) KCNH2DRD2HTR2A
Hydrochloric Acid SCHEMBL8566121 0.73 KCNH2 (0.76) KCNH2DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683782-A4 SPIRO (2H-1-BENZOPYRAN-2, 4' PIPERIDINE) CLASS III ANTIARRHYTHMICS. MERCK & CO INC (US) 1996-03-27 EP disclosed
EP-0683782-A1 SPIRO (2H-1-BENZOPYRAN-2, 4' PIPERIDINE) CLASS III ANTIARRHYTHMICS MERCK & CO. INC. (US) 1995-11-29 EP disclosed
WO-1994018204-A1 SPIRO (2H-1-BENZOPYRAN-2, 4' PIPERIDINE) CLASS III ANTIARRHYTHMICS MERCK & CO., INC. (US) 1994-08-18 WO disclosed