SCHEMBL9040482

SCHEMBL9040482

CN(CCc1c[nH]c2nc(N)nc(O)c12)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TYMS P04818 7/20 0.55
DHFR P00374 5/20 0.55
FOLR1 P15328 7/20 0.55
SLC19A1 P41440 6/20 0.55
SLC46A1 Q96NT5 6/20 0.55
GART P22102 2/20 0.53
FOLR2 P14207 2/20 0.48
EHMT2 Q96KQ7 1/20 0.48
ATIC P31939 1/20 0.46
SHMT1 P34896 1/20 0.46
FRK P42685 1/20 0.46
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9226749 0.97 FOLR1 (0.52) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9219313 0.97 FOLR1 (0.52) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9041174 0.93 DHFR (0.55) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9039369 0.88 TYMS (0.52) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL10448069 0.87 FOLR1 (0.51) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9224838 0.85 TYMS (0.49) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9228897 0.85 TYMS (0.49) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9439839 0.85 FOLR1 (0.74) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9227692 0.84 TYMS (0.50) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9691410 0.84 TYMS (0.50) TYMSDHFRFOLR1SLC19A1SLC46A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0400562-B1 Pyrrolopyrimidines, their production and use as tumoricidal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-08-21 EP disclosed