SCHEMBL904202

SCHEMBL904202

CS(=O)(=O)N1CCN(Cc2cc(F)c(O)c(F)c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
KDM4E B2RXH2 4/20 0.51
MAPT P10636 2/20 0.45
GAA P10253 2/20 0.45
POLB P06746 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CYP2D6 P10635 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
RECQL P46063 1/20 0.44
MAP4K4 O95819 1/20 0.43
LMNA P02545 1/20 0.43
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
HTT P42858 2/20 0.41
TSHR P16473 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL903893 0.84 ALDH1A1 (0.54) ALDH1A1KDM4ENPSR1SMN1; SMN2RECQL
SCHEMBL22683993 0.81 KDM4E (0.48) ALDH1A1KDM4ENPSR1CYP2D6SMN1; SMN2
SCHEMBL1003970 0.78 ALDH1A1 (0.51) ALDH1A1KDM4ENPSR1CYP2D6SMN1; SMN2
SCHEMBL17896800 0.78 MAP4K4 (0.50) ALDH1A1KDM4ENPSR1CYP2D6SMN1; SMN2
SCHEMBL940416 0.76 ALDH1A1 (0.62) ALDH1A1KDM4EMAPTNPSR1CYP2D6
SCHEMBL1005879 0.76 KDM4E (0.62) ALDH1A1KDM4ENPSR1CYP2D6SMN1; SMN2
SCHEMBL1006389 0.75 KDM4E (0.54) ALDH1A1KDM4ESMN1; SMN2LMNATSHR
SCHEMBL31010040 0.75 ALDH1A1 (0.62) ALDH1A1KDM4EGAAPOLBSMN1; SMN2
SCHEMBL2547164 0.74 KDM4E (0.53) ALDH1A1KDM4ENPSR1SMN1; SMN2RECQL
SCHEMBL17896323 0.74 KDM4E (0.50) ALDH1A1KDM4EPOLBNPSR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed