SCHEMBL9042575

SCHEMBL9042575

COC(=O)C(=O)c1ccc(OCCCC(O)c2ccc3ccccc3c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.51
HDAC8 Q9BY41 1/20 0.49
PPARG P37231 2/20 0.45
PPARD Q03181 2/20 0.45
PPARA Q07869 2/20 0.45
GABBR2 O75899 1/20 0.44
GABBR1 Q9UBS5 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
TSHR P16473 1/20 0.43
HIF1A Q16665 1/20 0.43
UTS2R Q9UKP6 2/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 1/20 0.42
AOC3 Q16853 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9042662 0.87 HDAC1 (0.51) HDAC1HDAC8PPARGPPARDPPARA
SCHEMBL9043319 0.84 HDAC1 (0.56) HDAC1HDAC8PPARGPPARDPPARA
SCHEMBL9041806 0.82 PPARG (0.59) HDAC1PPARGPPARDPPARAMEN1
SCHEMBL9042608 0.82 PPARA (0.38) HDAC1HDAC8PPARGPPARDPPARA
SCHEMBL9119262 0.81 MEN1 (0.47) HDAC1MEN1KMT2AMAPTRAB9A
SCHEMBL9042013 0.80 HDAC1 (0.52) HDAC1HDAC8PPARGPPARDPPARA
SCHEMBL9041562 0.80 PPARG (0.50) HDAC1HDAC8PPARGPPARDPPARA
SCHEMBL9043389 0.79 PPARG (0.54) HDAC1PPARGPPARDPPARAMAPT
SCHEMBL9045735 0.78 HDAC3 (0.55) HDAC1HDAC8MEN1KMT2ARAB9A
SCHEMBL9041688 0.78 CNR2 (0.50) HDAC1HDAC8PPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512352-B1 Substituted carboxylic acid derivatives HOFFMANN LA ROCHE (CH) 1996-03-27 EP disclosed
US-5344843-A Carnitine acryltransferase enzyme inhibitors as antiischemic agents and for cardiovascular disorders HOFFMAN-LA ROCHE INC. (US) 1994-09-06 US disclosed
EP-0512352-A2 Substituted carboxylic acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-11-11 EP disclosed