SCHEMBL9044792

SCHEMBL9044792

CCOC(=O)c1ccc(CCc2c[nH]c3nc(N)nc(O)c23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 4/20 0.51
DHFR P00374 4/20 0.51
NAMPT P43490 2/20 0.47
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAOA P21397 1/20 0.42
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ESR1 P03372 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
ESR2 Q92731 1/20 0.40
CA14 Q9ULX7 1/20 0.40
FOLR2 P14207 1/20 0.40
FOLR1 P15328 1/20 0.40
GART P22102 1/20 0.40
ATIC P31939 1/20 0.40
SHMT1 P34896 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047680 0.94 DHFR (0.45) TYMSDHFRNAMPTLMNACYP1A2
SCHEMBL7843188 0.90 NAMPT (0.57) TYMSDHFRNAMPTLMNACYP1A2
SCHEMBL14329878 0.90 DHFR (0.51) TYMSDHFRNAMPTCYP1A2CYP3A4
SCHEMBL9046718 0.85 TYMS (0.54) TYMSDHFRNAMPTFOLR2FOLR1
SCHEMBL15247798 0.84 NAMPT (0.52) TYMSDHFRNAMPTFOLR2FOLR1
SCHEMBL9044536 0.84 NAMPT (0.51) TYMSDHFRNAMPTLMNACYP1A2
SCHEMBL10306798 0.83 DHFR (0.48) TYMSDHFRNAMPTFOLR2FOLR1
SCHEMBL9042447 0.82 DHFR (0.64) TYMSDHFRNAMPTFOLR2FOLR1
SCHEMBL9042429 0.82 DHFR (0.64) TYMSDHFRNAMPTFOLR2FOLR1
SCHEMBL10306795 0.79 TYMS (0.58) TYMSDHFRNAMPTFOLR2FOLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549886-B1 Process for the preparation of pyrrolo[2,3-d]pyrimidines UNIV PRINCETON (US) 1996-10-30 EP disclosed
US-5254687-A Process for the preparation of pyrrolo[2,3-d]pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-10-19 US disclosed
EP-0549886-A1 Process for the preparation of pyrrolo[2,3-d]pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-07-07 EP disclosed