SCHEMBL9045812

SCHEMBL9045812

O=C(O)c1ccc2c(c1)OCc1ccccc1C2=CCCl

nearest known ligand 0.71

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 8/20 0.58
TBXAS1 P24557 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045798 1.00 TBXA2R (0.58) TBXA2RTBXAS1
SCHEMBL9044687 0.90 TBXA2R (0.67) TBXA2RTBXAS1
SCHEMBL9047398 0.90 TBXA2R (0.67) TBXA2RTBXAS1
SCHEMBL9044692 0.90 TBXA2R (0.67) TBXA2RTBXAS1
SCHEMBL9046600 0.89 TBXA2R (0.59) TBXA2RTBXAS1
SCHEMBL9046608 0.89 TBXA2R (0.59) TBXA2RTBXAS1
SCHEMBL8143121 0.84 TBXA2R (0.53) TBXA2RTBXAS1
SCHEMBL8143124 0.84 TBXA2R (0.53) TBXA2RTBXAS1
SCHEMBL5060505 0.83 HRH1 (0.69)
SCHEMBL5060502 0.83 HRH1 (0.69)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345747-B1 Tricyclic compounds KYOWA HAKKO KOGYO KK (JP) 1996-06-26 EP disclosed
US-5302596-A DIBENZO-CYCLOHEPTENES,-OXEPINS AND-THIEPINS SUBSTITUTED BY A HETEROCYCLO-ALKYL KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-04-12 US disclosed
US-5242931-A Antiischemic agents and cardiovascular disorders KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-07 US disclosed
US-5118701-A Antiischemic agents, anticoagulants KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-06-02 US disclosed
US-4999363-A Inhibit biosynthesis of thromboxane A2 KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-12 US disclosed
EP-0345747-A2 Tricyclic compounds KYOWA HAKKO KOGYO CO., LTD. (JP) 1989-12-13 EP disclosed