SCHEMBL9047220

SCHEMBL9047220

CC(C)(C)C(=O)c1c(CC(C)(C)C(=O)O)n(Cc2ccc(Cl)cc2)c2ccc(O)cc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 17/20 0.61
PTGES O14684 5/20 0.61
KDM4E B2RXH2 2/20 0.60
CYP1A2 P05177 2/20 0.60
CYP3A4 P08684 2/20 0.60
MAPT P10636 2/20 0.60
CYP2C9 P11712 2/20 0.60
HPGD P15428 2/20 0.60
HSD17B10 Q99714 2/20 0.60
TDP1 Q9NUW8 2/20 0.60
TSHR P16473 1/20 0.60
CYP2C19 P33261 1/20 0.60
HIF1A Q16665 1/20 0.60
ALOX5AP P20292 3/20 0.57
ALOX5 P09917 2/20 0.55
PTGS2 P35354 2/20 0.55
MEN1 O00255 1/20 0.55
USP2 O75604 1/20 0.55
TP53 P04637 1/20 0.55
POLB P06746 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562954 0.89 PTGES2 (0.57) PTGES2PTGESKDM4ECYP1A2CYP3A4
SCHEMBL23270737 0.89 PTGES2 (0.77) PTGES2PTGESKDM4ECYP1A2CYP3A4
SCHEMBL30181373 0.89 PTGES2 (0.77) PTGES2PTGESKDM4ECYP1A2CYP3A4
SCHEMBL9434490 0.87 PTGES2 (0.78) PTGES2PTGESKDM4ECYP1A2CYP3A4
SCHEMBL9736663 0.83 PTGES2 (0.61) PTGES2PTGESKDM4ECYP1A2CYP3A4
SCHEMBL9044519 0.82 ALOX5AP (0.79) PTGES2PTGESKDM4ECYP1A2CYP3A4
SCHEMBL9208334 0.81 PTGES2 (0.55) PTGES2PTGESKDM4ECYP1A2CYP3A4
SCHEMBL25968427 0.80 PTGES2 (0.66) PTGES2PTGESKDM4ECYP1A2CYP3A4
SCHEMBL9738077 0.79 PTGES2 (0.83) PTGES2PTGESKDM4ECYP1A2CYP3A4
SCHEMBL23270837 0.79 PTGES2 (0.64) PTGES2PTGESKDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0535925-B1 (Bicyclic-hetero-arylmethoxy)indoles as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC (CA) 1996-04-24 EP disclosed
US-5308850-A (Bicyclic-hetero-arylmethoxy)indoles as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1994-05-03 US disclosed
EP-0535925-A1 (Bicyclic-hetero-arylmethoxy)indoles as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1993-04-07 EP disclosed