SCHEMBL9047655

SCHEMBL9047655

COc1ncnc(N2CCC(N)C2)c1OC

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 4/20 0.51
DOT1L Q8TEK3 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
ACACB O00763 9/20 0.41
AKT2 P31751 4/20 0.41
LRRK2 Q5S007 1/20 0.40
KIT P10721 1/20 0.40
GSK3B P49841 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9049074 0.85 AKT1 (0.54) AKT1DOT1LHRH4AKT2LRRK2
SCHEMBL9048311 0.75 AKT1 (0.47) AKT1DOT1LHRH4AKT2LRRK2
SCHEMBL14599443 0.74 ENPP1 (0.67)
SCHEMBL9046030 0.74 HTR2C (0.44)
SCHEMBL16190458 0.69 ACACB (0.49) ACACB
SCHEMBL14275566 0.69 AKT1 (0.52) AKT1DOT1LHRH4AKT2KIT
SCHEMBL29364150 0.67 AKT1 (0.50) AKT1DOT1LHRH4AKT2
SCHEMBL23599086 0.67 NPC1 (0.63) AKT1DOT1LHRH4AKT2
SCHEMBL15178732 0.67 DOT1L (0.85) DOT1LAKT2KITGSK3B
SCHEMBL10074309 0.67 DOT1L (0.85) DOT1LAKT2KITGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714896-A1 INDOL DERIVATIVES USEFUL FOR THE TREATMENT OF MIGRAINE, COMPOSITION AND UTILIZATION VITA-INVEST, S.A. (ES) 1996-06-05 EP disclosed