SCHEMBL9047834

SCHEMBL9047834

c1ccc(CN2CCC(c3nc4c(s3)Cc3ccccc3-4)C2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.44
DAPK3 O43293 1/20 0.44
LTK P29376 1/20 0.44
MAPK8 P45983 1/20 0.44
CSNK1A1 P48729 1/20 0.44
CDK8 P49336 1/20 0.44
LIMK1 P53667 1/20 0.44
CDK5 Q00535 1/20 0.44
DYRK1A Q13627 1/20 0.44
LRRK2 Q5S007 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
DYRK1B Q9Y463 1/20 0.44
ADORA1 P30542 1/20 0.43
ACHE P22303 5/20 0.42
BCHE P06276 3/20 0.42
USP30 Q70CQ3 1/20 0.40
SIGMAR1 Q99720 2/20 0.40
DRD2 P14416 3/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9045678 0.99 ACHE (0.43) CHEK1DAPK3LTKMAPK8CSNK1A1
SCHEMBL9046905 0.81 ACHE (0.45) CHEK1DAPK3LTKMAPK8CSNK1A1
SCHEMBL9046200 0.81 CHEK1 (0.48) CHEK1DAPK3LTKMAPK8CSNK1A1
Hydrochloric Acid SCHEMBL9050349 0.80 ACHE (0.47) CHEK1DAPK3LTKMAPK8CSNK1A1
SCHEMBL9045402 0.78 CHEK1 (0.45) CHEK1DAPK3LTKMAPK8CSNK1A1
SCHEMBL9045662 0.78 BCHE (0.44) CHEK1DAPK3LTKMAPK8CSNK1A1
Hydrochloric Acid SCHEMBL9049947 0.76 BCHE (0.42) CHEK1DAPK3LTKMAPK8CSNK1A1
SCHEMBL9045761 0.74 CHEK1 (0.43) CHEK1DAPK3LTKMAPK8CSNK1A1
SCHEMBL9050942 0.74 CHEK1 (0.43) CHEK1DAPK3LTKMAPK8CSNK1A1
SCHEMBL9045403 0.74 CHEK1 (0.45) CHEK1DAPK3LTKMAPK8CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749966-A1 5-HT 3 RECEPTOR AGONIST, NOVEL THIAZOLE DERIVATIVE, AND INTERMEDIATE THEREFOR YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-12-27 EP disclosed