SCHEMBL9047895

SCHEMBL9047895

CCCCCCCCCCN1CCN(C(=O)OCC)CC1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 16/20 0.60
HRH1 P35367 16/20 0.60
ALDH1A1 P00352 1/20 0.50
POLB P06746 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
GAA P10253 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11747160 1.00 HRH2 (0.60) HRH2HRH1ALDH1A1POLBHTT
SCHEMBL27629332 0.98 HRH2 (0.59) HRH2HRH1ALDH1A1POLBHTT
SCHEMBL14670199 0.93 HRH2 (0.56) HRH2HRH1ALDH1A1POLBHTT
SCHEMBL15309235 0.88 HRH2 (0.52) HRH2HRH1ALDH1A1POLBHTT
SCHEMBL5540683 0.87 HRH2 (0.51) HRH2HRH1ALDH1A1POLBHTT
SCHEMBL27370873 0.86 HRH2 (0.57) HRH2HRH1
SCHEMBL9051052 0.85 ALDH1A1 (0.56) HRH2HRH1ALDH1A1POLBHTT
SCHEMBL11182660 0.85 HRH2 (0.52) HRH2HRH1ALDH1A1POLBHTT
SCHEMBL5542649 0.85 HRH2 (0.52) HRH2HRH1ALDH1A1POLBHTT
SCHEMBL11392680 0.84 HRH2 (0.55) HRH2HRH1ALDH1A1POLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0703908-A1 ANALGESIC DIBENZOXAZEPINES AND DIBENZOTHIAZEPINES G.D. SEARLE & CO. (US) 1996-04-03 EP disclosed
US-5461047-A Analgesics and treats prostaglandin-E2 mediated diseases in animals G. D. SEARLE & CO. (US) 1995-10-24 US disclosed
WO-1994029286-A1 ANALGESIC DIBENZOXAZEPINES AND DIBENZOTHIAZEPINES G.D. SEARLE & CO. (US) 1994-12-22 WO disclosed
US-5354747-A Analgesics G. D. SEARLE & CO. (US) 1994-10-11 US disclosed
US-4036828-A 3,4-Bis(4-substituted piperazinyl)-3-cyclobutene-1,2-diones and related compounds G. D. SEARLE & CO. (US) 1977-07-19 US disclosed