SCHEMBL9048449

SCHEMBL9048449

CC(OCC(O)c1cccc2ccccc12)c1cnc[nH]1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 13/20 0.64
ADRA2B P18089 13/20 0.64
ADRA2C P18825 13/20 0.64
ADRA1A P35348 9/20 0.64
ADRA1B P35368 8/20 0.64
ADRA1D P25100 7/20 0.64
KCNH2 Q12809 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
SLC6A2 P23975 1/20 0.41
HTR7 P34969 1/20 0.41
CASR P41180 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21401251 0.79 ADRA2A (1.00) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL21401258 0.77 ADRA2A (1.00) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL31578481 0.77 ADRA2A (1.00) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL8478307 0.77 ADRA2A (0.54) ADRA2AADRA2BADRA2CADRA1AADRA1B
Hydrochloric Acid SCHEMBL29368290 0.76 ADRA2A (0.97) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL9255140 0.75 ADRA2A (0.52) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL21401252 0.74 ADRA2A (1.00) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL2626829 0.74 ADRA2A (0.68) ADRA2AADRA2BADRA2CADRA1AADRA1B
Hydrochloric Acid SCHEMBL8480333 0.71 TSHR (0.42) ADRA2AADRA2CADRA1AKCNH2TP53
Hydrochloric Acid SCHEMBL8482510 0.71 AOC3 (0.43) ADRA2AADRA2BADRA2CTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0589484-B1 1,2-Ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same TOYAMA CHEMICAL CO LTD (JP) 1996-10-16 EP claimed
EP-0589484-A1 1,2-Ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same TOYAMA CHEMICAL CO., LTD. (JP) 1994-03-30 EP claimed
EP-0383281-A1 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same TOYAMA CHEMICAL CO., LTD. (JP) 1990-08-22 EP claimed
US-5472984-A 1,2-ethanediol derivative and salt thereof and cerebral function-improving agent comprising the same TOYAMA CHEMICAL CO., LTD. (JP) 1995-12-05 US disclosed