SCHEMBL9051214

SCHEMBL9051214

CCCCNC(=O)[C@@H]1C[C@H](Oc2ccccc2)CN1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.43
PRCP P42785 2/20 0.42
CTSC P53634 1/20 0.42
HPGD P15428 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
TLR2 O60603 3/20 0.40
TLR1 Q15399 3/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
BCHE P06276 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL9595917 0.94 CTSC (0.40) HRH3PRCPCTSCHPGDMAPT
Trifluoroacetic Acid SCHEMBL9054201 0.79 NCEH1 (0.38) CTSCHPGD
SCHEMBL6412333 0.78 L3MBTL1 (0.47) HRH3CTSC
SCHEMBL951361 0.77 HRH3 (0.50) HRH3CTSCHPGDMAPT
SCHEMBL3961763 0.77 HRH3 (0.50) HRH3CTSCHPGDMAPT
SCHEMBL23260557 0.77 HRH3 (0.50) HRH3CTSCHPGDMAPT
SCHEMBL950955 0.77 HRH3 (0.50) HRH3CTSCHPGDMAPT
SCHEMBL7733533 0.77 EPHX2 (0.40) HRH3
SCHEMBL464484 0.76 HRH3 (0.52) HRH3
SCHEMBL14037635 0.76 HRH3 (0.52) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696277-A1 HIV PROTEASE INHIBITORS USEFUL FOR THE TREATMENT OF AIDS MERCK & CO. INC. (US) 1996-02-14 EP disclosed
WO-1994022480-A1 HIV PROTEASE INHIBITORS IN PHARMACEUTICAL COMBINATIONS FOR THE TREATMENT OF AIDS MERCK & CO., INC. (US) 1994-10-13 WO disclosed