SCHEMBL9051277

SCHEMBL9051277

O=C1N=CCOc2c1oc1cc(Cl)ccc21

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.37
TTR P02766 2/20 0.37
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
MKNK2 Q9HBH9 1/20 0.36
DAO P14920 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
MCL1 Q07820 1/20 0.35
CDC25A P30304 1/20 0.34
CDC25C P30307 1/20 0.34
ADORA3 P0DMS8 2/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
AKR1B1 P15121 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
ALPL P05186 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6650554 0.69 DAO (0.39) AHRTTRCA1CA2MKNK2
SCHEMBL11728871 0.64 TTR (0.71) AHRTTRCA1CA2DAO
SCHEMBL29465920 0.64 TTR (0.71) AHRTTRCA1CA2DAO
SCHEMBL6678399 0.64 ALPL (0.39) TTRCA1CA2DAOMCL1
SCHEMBL5378213 0.63 TTR (0.51) AHRTTRCA1CA2DAO
SCHEMBL15842804 0.63 AHR (0.50) AHRTTRCA1CA2DAO
SCHEMBL22737968 0.63 AHR (0.78) AHRTTRCA1CA2DAO
SCHEMBL29908973 0.62 TTR (0.54) AHRTTRCA1CA2CYP11B1
SCHEMBL27244495 0.62 TTR (0.54) AHRTTRCA1CA2CYP11B1
SCHEMBL15842242 0.60 KDM4E (0.57) AHRTTRCA1CA2DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749434-A1 BENZOTHIOPHENE, BENZOFURAN AND INDOLETHIAZEPINONES, OXAZEPINONES AND DIAZEPINONES AS INHIBITORS OF CELL ADHESION AND AS INHIBITORS OF HIV WARNER-LAMBERT COMPANY (US) 1996-12-27 EP disclosed
WO-1995024408-A1 BENZOTHIOPHENE, BENZOFURAN AND INDOLETHIAZEPINONES, OXAZEPINONES AND DIAZEPINONES AS INHIBITORS OF CELL ADHESION AND AS INHIBITORS OF HIV WARNER-LAMBERT COMPANY (US) 1995-09-14 WO disclosed