SCHEMBL9053085

SCHEMBL9053085

COc1ccc(-c2cc(C#N)nn2-c2ccc(S(N)(=O)=O)cc2)cc1Br.N#Cc1cc(-c2ccccc2)n(-c2ccc(S(N)(=O)=O)cc2)n1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.62
CYP2C9 P11712 1/20 0.52
PTGS1 P23219 7/20 0.52
ABCB11 O95342 1/20 0.51
ALDH1A1 P00352 1/20 0.51
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
CA9 Q16790 3/20 0.50
PDPK1 O15530 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6340631 0.95 PTGS2 (0.65) PTGS2PTGS1ABCB11ALDH1A1CA1
SCHEMBL9053327 0.93 PTGS2 (0.55) PTGS2CYP2C9PTGS1ABCB11ALDH1A1
SCHEMBL6341657 0.86 PTGS2 (0.78) PTGS2CYP2C9PTGS1CA1CA2
SCHEMBL6341186 0.84 PTGS2 (0.69) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6340846 0.84 PTGS2 (0.75) PTGS2PTGS1CA1CA2CA9
SCHEMBL7867795 0.83 PTGS2 (0.53) PTGS2CYP2C9PTGS1
SCHEMBL8689101 0.82 PTGS2 (0.42) PTGS2PTGS1ABCB11ALDH1A1CA1
SCHEMBL6341745 0.81 PTGS2 (0.78) PTGS2CYP2C9PTGS1CA1CA2
SCHEMBL6350193 0.79 PTGS2 (0.78) PTGS2CYP2C9PTGS1ABCB11CA1
SCHEMBL17456918 0.78 PTGS2 (0.75) PTGS2CYP2C9PTGS1ABCB11CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731795-A1 SUBSTITUTED PYRAZOLYL BENZENESULFONAMIDES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP claimed