SCHEMBL9053306

SCHEMBL9053306

CCOC(=O)c1ccc(N=Cc2ccc3c(c2)OCCC3(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
HPGD P15428 3/20 0.47
KDM4E B2RXH2 2/20 0.47
TSHR P16473 1/20 0.47
RARA P10276 7/20 0.46
RARB P10826 7/20 0.46
RARG P13631 4/20 0.46
RXRA P19793 2/20 0.43
HNF4A P41235 1/20 0.43
MAPT P10636 4/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
GAA P10253 1/20 0.40
F2 P00734 1/20 0.40
HIF1A Q16665 1/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9093004 0.92 RARB (0.53) ALDH1A1HPGDKDM4ETSHRRARA
SCHEMBL9091706 0.85 RARB (0.56) ALDH1A1KDM4ERARARARBRARG
SCHEMBL9053667 0.85 ALDH1A1 (0.52) ALDH1A1HPGDKDM4ETSHRRARA
SCHEMBL9054214 0.84 ALDH1A1 (0.47) ALDH1A1HPGDKDM4ETSHRRARA
SCHEMBL9143040 0.82 RARB (0.66) ALDH1A1KDM4ERARARARBRARG
SCHEMBL9143045 0.82 RARB (0.66) ALDH1A1KDM4ERARARARBRARG
SCHEMBL9053417 0.81 ALDH1A1 (0.48) ALDH1A1HPGDKDM4ETSHRRARA
SCHEMBL9057342 0.80 ALDH1A1 (0.47) ALDH1A1HPGDKDM4ETSHRRARA
SCHEMBL11597612 0.80 MAPT (0.60) ALDH1A1HPGDKDM4ETSHRMAPT
SCHEMBL11597609 0.80 MAPT (0.60) ALDH1A1HPGDKDM4ETSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5498755-A IMINE COMPOUNDS FOR SKIN DISORDERS AND ANTIINFLAMMATORY AGENTS ALLERGAN, INC. 1996-03-12 US disclosed
WO-1996006070-A1 DISUBSTITUTED ARYL AND HETEROARYL IMINES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1996-02-29 WO disclosed