SCHEMBL9053674

SCHEMBL9053674

O=C(O)CSc1nnc(SSc2nnc(SCC(=O)O)s2)s1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.67
L3MBTL1 Q9Y468 2/20 0.67
APEX1 P27695 1/20 0.57
HPGD P15428 4/20 0.51
ALDH1A1 P00352 4/20 0.51
POLB P06746 3/20 0.51
FFAR1 O14842 2/20 0.51
KDM4E B2RXH2 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
MEN1 O00255 1/20 0.44
ESR1 P03372 1/20 0.44
TSHR P16473 1/20 0.44
RECQL P46063 1/20 0.44
BLM P54132 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8436040 0.94 GAA (0.74) GAAL3MBTL1APEX1HPGDALDH1A1
SCHEMBL14384511 0.84 GAA (0.62) GAAL3MBTL1APEX1HPGDALDH1A1
SCHEMBL14557231 0.84 GAA (0.68) GAAL3MBTL1APEX1HPGDALDH1A1
SCHEMBL14582756 0.84 GAA (0.62) GAAL3MBTL1APEX1HPGDALDH1A1
SCHEMBL11860585 0.82 GAA (0.66) GAAL3MBTL1APEX1HPGDALDH1A1
SCHEMBL11499467 0.82 GAA (0.56) GAAL3MBTL1APEX1HPGDALDH1A1
SCHEMBL8441615 0.81 GAA (0.48) GAAL3MBTL1APEX1HPGDALDH1A1
SCHEMBL1964151 0.80 L3MBTL1 (0.62) GAAL3MBTL1APEX1HPGDALDH1A1
SCHEMBL9443307 0.80 GAA (0.62) GAAL3MBTL1APEX1HPGDALDH1A1
SCHEMBL1686848 0.80 GAA (1.00) GAAL3MBTL1HPGDALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996007676-A1 POLYMERIC RESIN FOR DISULFIDE BOND SYNTHESIS EKAGEN CORPORATION (US) 1996-03-14 WO disclosed
EP-0194571-B1 HETEROCYCLIC DISULFIDES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1990-11-14 EP disclosed
US-4656262-A 7-methoxy cephalosporin derivative YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1987-04-07 US disclosed
EP-0194571-A1 Heterocyclic disulfides, process for their preparation and pharmaceutical preparations containing them HOECHST AKTIENGESELLSCHAFT (DE) 1986-09-17 EP disclosed
US-4242449-A 7-Methoxy cephalosporins and process of producing them YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1980-12-30 US disclosed