SCHEMBL9056570

SCHEMBL9056570

Cn1cc(CCNc2cccnc2)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.51
HTR2A P28223 1/20 0.50
GPR84 Q9NQS5 1/20 0.48
SPR P35270 1/20 0.45
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
HTR6 P50406 1/20 0.44
CDK2 P24941 1/20 0.43
IP6K1 Q92551 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CA2 P00918 1/20 0.41
HDAC3 O15379 2/20 0.41
HDAC4 P56524 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC7 Q8WUI4 2/20 0.41
HDAC2 Q92769 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9054532 0.93 HTR2C (0.49) HTR2CHTR2AGPR84KEAP1NFE2L2
Maleic Acid SCHEMBL8415335 0.84 MEN1 (0.48) HTR2CCDK2MEN1KMT2AKDM4E
Fumaric Acid SCHEMBL8415339 0.84 MEN1 (0.48) HTR2CCDK2MEN1KMT2AKDM4E
SCHEMBL9055209 0.81 HTR2C (0.79) HTR2CHTR6KMT2ALMNA
SCHEMBL8804198 0.80 NOTUM (0.62) MEN1KMT2AKDM4EHPGDHSD17B10
SCHEMBL14817117 0.79 TP53 (0.55) HTR2AGPR84KEAP1NFE2L2HTR6
SCHEMBL8418207 0.78 HTR2A (0.51) HTR2AGPR84KEAP1NFE2L2HTR6
SCHEMBL8415790 0.78 HTR2C (0.67) HTR2CHTR6MEN1KMT2ARXFP1
SCHEMBL8265671 0.77 HTR2A (0.61) HTR2AGPR84KEAP1NFE2L2HTR6
SCHEMBL8804773 0.77 PTPN5 (0.64) MEN1KMT2AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004266-A2 INDOL, INDAZOL, PYRIDOPYRROL AND PYRIDOPYRAZOL DERIVATIVES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY AND IMMUNOMODULATING EFFECTS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1996-02-15 WO disclosed