SCHEMBL8418207

SCHEMBL8418207

Cn1cc(CCCNc2ccncc2)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.51
GPR84 Q9NQS5 1/20 0.49
KDM4E B2RXH2 2/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HPGD P15428 1/20 0.48
HSD17B10 Q99714 1/20 0.48
LMNA P02545 3/20 0.46
RXFP1 Q9HBX9 2/20 0.46
TP53 P04637 2/20 0.46
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
SLC6A2 P23975 1/20 0.44
HTR6 P50406 1/20 0.42
CA2 P00918 1/20 0.42
SLC6A4 P31645 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9054532 0.86 HTR2C (0.49) HTR2AGPR84KDM4EMEN1KMT2A
Maleic Acid SCHEMBL8415335 0.78 MEN1 (0.48) KDM4EMEN1KMT2AHPGDHSD17B10
Fumaric Acid SCHEMBL8415339 0.78 MEN1 (0.48) KDM4EMEN1KMT2AHPGDHSD17B10
SCHEMBL9056570 0.78 HTR2C (0.51) HTR2AGPR84KDM4EMEN1KMT2A
SCHEMBL7004405 0.78 HTR2A (0.73) HTR2AGPR84KDM4EMEN1KMT2A
SCHEMBL9055889 0.78 DNM2 (0.47) KDM4EHSD17B10TP53SLC6A2HTR6
SCHEMBL6351593 0.77 HTR2A (0.59) HTR2AGPR84KDM4EMEN1KMT2A
SCHEMBL8418107 0.77 CYP19A1 (0.56) MEN1KMT2ARXFP1HTR6ALDH1A1
SCHEMBL14817117 0.77 TP53 (0.55) HTR2AGPR84KDM4EMEN1KMT2A
SCHEMBL5096037 0.77 GSK3B (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965582-A ANTIHISTAMINES ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1999-10-12 US claimed
WO-1996004266-A2 INDOL, INDAZOL, PYRIDOPYRROL AND PYRIDOPYRAZOL DERIVATIVES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY AND IMMUNOMODULATING EFFECTS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1996-02-15 WO claimed