SCHEMBL9058573

SCHEMBL9058573

O=[N+]([O-])c1cnc2ccc[c]n12

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALDH1A1 P00352 3/20 0.36
GAA P10253 1/20 0.36
LMNA P02545 3/20 0.33
MAPK1 P28482 2/20 0.33
THRB P10828 2/20 0.33
TSHR P16473 1/20 0.33
ATM Q13315 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CHRM1 P11229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29018907 0.69 CYP1A2 (0.57) CYP1A2CYP2C9ALDH1A1LMNAMEN1
SCHEMBL7998162 0.68 MKNK1 (0.46) CYP1A2CYP2C9ALDH1A1GAALMNA
SCHEMBL6743031 0.67 CYP1A2 (0.43) CYP1A2CYP2C9ALDH1A1GAALMNA
SCHEMBL9001950 0.67 ATM (0.46) CYP1A2CYP2C9ALDH1A1GAALMNA
SCHEMBL6742620 0.67 CYP1A2 (0.54) CYP1A2CYP2C9ALDH1A1GAALMNA
SCHEMBL6746118 0.61 CYP1A2 (0.41) CYP1A2CYP2C9ALDH1A1GAALMNA
SCHEMBL20125049 0.60 CYP1A2 (1.00) CYP1A2CYP2C9ALDH1A1GAALMNA
SCHEMBL6742637 0.60 CYP1A2 (0.40) CYP1A2CYP2C9ALDH1A1GAALMNA
SCHEMBL430605 0.60 TNF (0.50) CYP1A2CYP2C9ALDH1A1GAAKDM4E
SCHEMBL28921245 0.60 CYP1A2 (0.67) CYP1A2CYP2C9ALDH1A1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632040-A1 Antibacterial imidazole derivatives Takeda Chemical Industries, Ltd. (JP) 1995-01-04 EP claimed
WO-1996016656-A1 CONDENSED IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-06 WO disclosed
EP-0632040-A1 Antibacterial imidazole derivatives Takeda Chemical Industries, Ltd. (JP) 1995-01-04 EP disclosed