SCHEMBL9060653

SCHEMBL9060653

CCc1ccc(/C=C/c2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
TUBB1 Q9H4B7 1/20 0.47
ALOX5 P09917 1/20 0.46
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAOB P27338 1/20 0.44
SLC6A4 P31645 1/20 0.43
CYP2D6 P10635 1/20 0.42
POLB P06746 1/20 0.42
KDM1A O60341 1/20 0.42
RCOR1 Q9UKL0 1/20 0.42
RELA Q04206 1/20 0.42
GRIK1 P39086 1/20 0.42
GRIK2 Q13002 1/20 0.42
PPARG P37231 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9060664 1.00 TSHR (0.49) TSHRTUBB1ALOX5PTGS1PTGS2
SCHEMBL155707 0.88 TSHR (0.58) TSHRALDH1A1LMNAMAPTSLC6A4
SCHEMBL9060735 0.88 TSHR (0.45) TSHRALDH1A1LMNASLC6A4CYP2D6
SCHEMBL9060736 0.88 TSHR (0.45) TSHRALDH1A1LMNASLC6A4CYP2D6
Ammonia Solution, Strong SCHEMBL25380785 0.86 TSHR (0.56) TSHRALDH1A1LMNAMAPTSMN1; SMN2
SCHEMBL13790221 0.86 CYP2D6 (0.50) PTGS1MAPTMAOBCYP2D6RELA
SCHEMBL9061030 0.85 PPARG (0.46) TSHRALOX5ALDH1A1SLC6A4PPARG
SCHEMBL9061019 0.85 PPARG (0.46) TSHRALOX5ALDH1A1SLC6A4PPARG
SCHEMBL7788592 0.84 TSHR (0.45) TSHRALDH1A1LMNAMAPTHPGD
SCHEMBL7788596 0.84 TSHR (0.45) TSHRALDH1A1LMNAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536442-A ELECTROOPTICS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-07-16 US disclosed
US-5324449-A Substituted phenyl trifluoromethyl ethers MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-06-28 US disclosed
EP-0334911-B1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1993-02-10 EP disclosed
EP-0334911-A1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1989-10-04 EP disclosed