SCHEMBL9060735

SCHEMBL9060735

CCCc1ccc(/C=C/c2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
SLC6A4 P31645 5/20 0.43
SLC6A3 Q01959 4/20 0.43
PPARG P37231 3/20 0.43
PPARA Q07869 3/20 0.43
GPR84 Q9NQS5 1/20 0.43
ALDH1A1 P00352 1/20 0.42
THRB P10828 1/20 0.41
DAO P14920 1/20 0.41
LMNA P02545 1/20 0.41
CYP2D6 P10635 1/20 0.40
GRIK1 P39086 1/20 0.39
GRIK2 Q13002 1/20 0.39
POLB P06746 1/20 0.39
KDM1A O60341 1/20 0.39
RCOR1 Q9UKL0 1/20 0.39
RELA Q04206 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9060736 1.00 TSHR (0.45) TSHRSLC6A4SLC6A3PPARGPPARA
SCHEMBL9061030 0.90 PPARG (0.46) TSHRSLC6A4SLC6A3PPARGPPARA
SCHEMBL9061019 0.90 PPARG (0.46) TSHRSLC6A4SLC6A3PPARGPPARA
SCHEMBL1687455 0.89 TSHR (0.53) TSHRSLC6A4SLC6A3GPR84ALDH1A1
SCHEMBL9061347 0.89 FAAH (0.47) TSHRSLC6A4SLC6A3PPARGPPARA
SCHEMBL9061353 0.89 FAAH (0.47) TSHRSLC6A4SLC6A3PPARGPPARA
SCHEMBL9060653 0.88 TSHR (0.49) TSHRSLC6A4PPARGPPARAALDH1A1
SCHEMBL9060664 0.88 TSHR (0.49) TSHRSLC6A4PPARGPPARAALDH1A1
SCHEMBL9062000 0.88 FAAH (0.49) TSHRSLC6A4SLC6A3PPARGPPARA
SCHEMBL9060456 0.88 FAAH (0.49) TSHRSLC6A4SLC6A3PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536442-A ELECTROOPTICS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-07-16 US disclosed
US-5324449-A Substituted phenyl trifluoromethyl ethers MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-06-28 US disclosed
EP-0334911-B1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1993-02-10 EP disclosed
EP-0334911-A1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1989-10-04 EP disclosed