SCHEMBL9063402

SCHEMBL9063402

C[C@@H](O)/C=C/c1cccc(-c2ccc(C#N)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.41
CYP11B2 P19099 1/20 0.40
MMP3 P08254 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
HDAC2 Q92769 3/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
XDH P47989 1/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
HSD11B1 P28845 3/20 0.37
ADAMTS4 O75173 1/20 0.37
MMP12 P39900 1/20 0.36
MMP13 P45452 1/20 0.36
KAT6A Q92794 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
MMP2 P08253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9063404 1.00 PTGS2 (0.41) PTGS2CYP11B2MMP3HRH3HDAC2
SCHEMBL9064292 0.86 HDAC2 (0.43) PTGS2MMP3HRH3HDAC2XDH
SCHEMBL9065315 0.81 BCL2L1 (0.50) PTGS2HDAC2HDAC8
SCHEMBL9063938 0.81 BCL2L1 (0.50) PTGS2HDAC2HDAC8
SCHEMBL9063368 0.81 PTGS2 (0.43) PTGS2HDAC2HDAC8
SCHEMBL9064317 0.81 BCL2L1 (0.50) PTGS2HDAC2HDAC8
SCHEMBL9063633 0.81 BCL2L1 (0.50) PTGS2HDAC2HDAC8
SCHEMBL9063991 0.81 PTGS2 (0.43) PTGS2HDAC2HDAC8
SCHEMBL9063937 0.81 BCL2L1 (0.50) PTGS2HDAC2HDAC8
SCHEMBL9064312 0.81 BCL2L1 (0.50) PTGS2HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696272-A1 CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITING N(3-BIPHENYLYL-1(S)-METHYL-2-PROPENYL) ACETOHYDROXAMIC ACID DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1996-02-14 EP disclosed
WO-1994025431-A1 CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITING N(3-BIPHENYLYL-1(S)-METHYL-2-PROPENYL) ACETOHYDROXAMIC ACID DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1994-11-10 WO disclosed