Bromide

Bromide

SCHEMBL9070504

Br.O.Oc1ccc2nccc(NC3CCCCC3)c2c1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT5B Q4FZB7 2/20 0.59
KMT5C Q86Y97 2/20 0.59
S1PR1 P21453 2/20 0.44
S1PR3 Q99500 1/20 0.44
IDO1 P14902 1/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 1/20 0.43
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
RIPK2 O43353 2/20 0.40
KDR P35968 2/20 0.40
NSD2 O96028 1/20 0.40
DYRK1A Q13627 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
IP6K1 Q92551 1/20 0.40
MAPK10 P53779 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9073082 0.97 KMT5B (0.62) KMT5BKMT5CS1PR1S1PR3IDO1
SCHEMBL30307410 0.77 KMT5B (0.62) KMT5BKMT5CS1PR1S1PR3IDO1
SCHEMBL17241563 0.76 KMT5B (0.59) KMT5BKMT5CCYP2D6CYP2C19KDM4E
Hydrochloric Acid SCHEMBL9070436 0.75 KDM4E (0.55) KMT5BKMT5CS1PR1IDO1CYP2D6
SCHEMBL529480 0.74 MELK (0.59) KMT5BKMT5CDYRK1ADYRK1BMAPKAPK2
SCHEMBL529479 0.74 MELK (0.59) KMT5BKMT5CDYRK1ADYRK1BMAPKAPK2
SCHEMBL2621803 0.73 SLC22A12 (0.55) KMT5BKMT5CCYP2D6CYP2C19KDM4E
SCHEMBL12871473 0.72 KMT5B (0.97) KMT5BKMT5CCYP2D6CYP2C19KDM4E
SCHEMBL9069386 0.70 SYK (0.48) RIPK2KDRMAPK14RETMAPKAPK2
SCHEMBL6071399 0.70 KMT5B (0.52) KMT5BKMT5CCYP2D6NSD2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5506235-A Quinoline derivatives as immunostimulants PFIZER INC. (US) 1996-04-09 US disclosed