SCHEMBL907627

SCHEMBL907627

CC(C)(C)[Si](C)(C)O[C@H](c1ccccc1)C1CCC(Cc2ccc(N)cc2)N1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.32
SIGMAR1 Q99720 1/20 0.30
SOAT1 P35610 1/20 0.30
DAGLA Q9Y4D2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11904856 1.00 OPRK1 (0.32) OPRK1SIGMAR1SOAT1DAGLA
SCHEMBL11928190 1.00 OPRK1 (0.32) OPRK1SIGMAR1SOAT1DAGLA
SCHEMBL11928235 1.00 OPRK1 (0.32) OPRK1SIGMAR1SOAT1DAGLA
SCHEMBL907628 1.00 OPRK1 (0.32) OPRK1SIGMAR1SOAT1DAGLA
SCHEMBL11928189 1.00 OPRK1 (0.32) OPRK1SIGMAR1SOAT1DAGLA
SCHEMBL13269859 0.91 SLC6A4 (0.33)
SCHEMBL13269858 0.91 SLC6A4 (0.33)
SCHEMBL1728506 0.91 CETP (0.34)
SCHEMBL1200502 0.91 CETP (0.34)
SCHEMBL1199605 0.91 CETP (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276756-B9 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME (US) 2012-08-15 EP disclosed
WO-2012010862-A3 IMPROVED COMBUSTIBLE COMPOSITION RECKITT BENCKISER SOUTH AFRICA (PTY) LIMITED (ZA) 2012-05-10 WO disclosed
EP-2276756-A1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS Merck Sharp & Dohme Corp. (US) 2011-01-26 EP disclosed