SCHEMBL9080571

SCHEMBL9080571

CCN(Cc1ccc(S(=O)(=O)c2ccccc2)cc1)c1ccc2c3c(cccc13)C(=O)N2

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 5/20 0.79
KDM4E B2RXH2 8/20 0.50
ALDH1A1 P00352 6/20 0.50
HPGD P15428 4/20 0.50
HSD17B10 Q99714 4/20 0.50
CASP1 P29466 3/20 0.50
CASP7 P55210 3/20 0.50
HTT P42858 2/20 0.50
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
POLB P06746 3/20 0.44
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PTPRB P23467 1/20 0.43
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9702076 0.89 TYMS (0.75) TYMSKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9508657 0.89 TYMS (0.63) TYMSKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9080093 0.89 TYMS (1.00) TYMSKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9508016 0.77 TYMS (0.58) TYMS
SCHEMBL9704001 0.74 TYMS (0.62) TYMSKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9504724 0.74 TYMS (0.52) TYMS
SCHEMBL9704015 0.73 TYMS (0.67) TYMSKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9506816 0.69 TYMS (0.62) TYMSKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9701868 0.69 TYMS (0.76) TYMSKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9702062 0.68 TYMS (0.61) TYMSKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5574039-A ANTITUMOR, FUNGICIDES AGOURON PHARMACEUTICALS, INC. (US) 1996-11-12 US disclosed
EP-0550566-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS (US) 1993-07-14 EP disclosed
WO-1992005153-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1992-04-02 WO disclosed