SCHEMBL9702062

SCHEMBL9702062

O=C1Nc2ccc(N(CCCO)Cc3ccc(S(=O)(=O)NN4CCNCC4)cc3)c3cccc1c23

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 4/20 0.61
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
BRD4 O60885 1/20 0.39
KLK7 P49862 1/20 0.38
KDM4E B2RXH2 7/20 0.37
ALDH1A1 P00352 7/20 0.37
PTPRB P23467 1/20 0.37
POLB P06746 3/20 0.37
ALPL P05186 1/20 0.37
HPGD P15428 5/20 0.36
CASP1 P29466 3/20 0.36
CASP7 P55210 3/20 0.36
HSD17B10 Q99714 3/20 0.36
TSHR P16473 2/20 0.36
USP2 O75604 1/20 0.36
ALOX15 P16050 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
CDK5 Q00535 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9506816 0.95 TYMS (0.62) TYMSMEN1KMT2ABRD4KLK7
SCHEMBL9704015 0.90 TYMS (0.67) TYMSMEN1KMT2ABRD4KLK7
SCHEMBL9701868 0.86 TYMS (0.76) TYMSBRD4KLK7KDM4EALDH1A1
SCHEMBL9703980 0.84 TYMS (0.62) TYMSBRD4KLK7KDM4EALDH1A1
SCHEMBL9080571 0.68 TYMS (0.79) TYMSMEN1KMT2ABRD4KLK7
SCHEMBL9702076 0.66 TYMS (0.75) TYMSMEN1KMT2ABRD4KLK7
SCHEMBL9080093 0.65 TYMS (1.00) TYMSMEN1KMT2ABRD4KLK7
SCHEMBL9504689 0.62 ALDH1A1 (0.47) MEN1KMT2ABRD4KDM4EALDH1A1
SCHEMBL29774550 0.60 TYMS (0.48) TYMSMEN1KMT2AKDM4EALDH1A1
SCHEMBL22533183 0.60 TYMS (0.48) TYMSMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992005153-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1992-04-02 WO disclosed