Razoxane

Razoxane

SCHEMBL9089

CC(CN1CC(=O)NC(=O)C1)N1CC(=O)NC(=O)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TOP2ATOP2B

The experimentally established mechanism targets of Razoxane. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TOP2A known ✓ P11388 3/20 1.00
TOP2B known ✓ Q02880 3/20 1.00
PTGS1 P23219 2/20 1.00
LMNA P02545 1/20 1.00
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
CRBN Q96SW2 1/20 0.35
PIK3CD O00329 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dexrazoxane SCHEMBL18400 1.00 TOP2A (1.00) TOP2ATOP2BPTGS1LMNAALDH1A1
Dexrazoxane SCHEMBL1586271 1.00 TOP2A (1.00) TOP2ATOP2BPTGS1LMNAALDH1A1
Razoxane SCHEMBL27174203 0.98 TOP2A (0.96) TOP2ATOP2BPTGS1LMNAALDH1A1
Razoxane SCHEMBL27748349 0.98 TOP2A (0.96) TOP2ATOP2BPTGS1LMNAALDH1A1
Dexrazoxane SCHEMBL18188 0.98 TOP2A (0.96) TOP2ATOP2BPTGS1LMNAALDH1A1
Dexrazoxane SCHEMBL18189 0.96 TOP2A (0.93) TOP2ATOP2BPTGS1LMNAALDH1A1
Dexrazoxane SCHEMBL27918475 0.96 TOP2A (0.93) TOP2ATOP2BPTGS1LMNAALDH1A1
Dexrazoxane SCHEMBL28086609 0.94 TOP2A (0.89) TOP2ATOP2BPTGS1LMNAALDH1A1
Dexrazoxane SCHEMBL5488431 0.91 TOP2A (0.83) TOP2ATOP2BPTGS1LMNAALDH1A1
Dexrazoxane SCHEMBL5295434 0.91 TOP2A (0.83) TOP2ATOP2BPTGS1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 29832 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748859-A2 CHEMICALLY AND PHOTOCHEMICALLY INITIATED CELL MEMBRANE BLEBBING TO INDUCE CELL VESICLE PRODUCTION, MODIFICATIONS THEREOF, AND USES THEREOF The Regents of the University of California (US) 2026-05-27 EP claimed
US-20260137794-A1 LIGAND-DRUG CONJUGATE AND USE THEREOF SYSTIMMUNE INC (US) 2026-05-21 US claimed
EP-4743490-A1 HUMANIZED ANTI-CD7 ANTIBODY Christian-Albrechts-Universität zu Kiel (DE) 2026-05-20 EP claimed
WO-2026099502-A1 NOVEL DRUG CONJUGATES FOR TESTING CELLULAR DRUG UPTAKE Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2026-05-15 WO claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
US-20260085100-A1 METHODS OF ANTIGEN PRODUCTION THE WISTAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2026-03-26 US claimed
US-12577255-B2 MDM2-based modulators of proteolysis and associated methods of use ARVINAS OPERATIONS, INC. (US) 2026-03-17 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
EP-4704832-A2 BIFUNCTIONAL SMALL MOLECULES TO TARGET THE SELECTIVE DEGRADATION OF CIRCULATING PROTEINS Biohaven Therapeutics Ltd. (VG) 2026-03-11 EP claimed
EP-4698185-A1 METHODS AND SYSTEMS FOR IMPROVING ANTI-CANCER THERAPIES Osasuna Therapeutics SA (CH) 2026-02-25 EP claimed
EP-0393575-B1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent SEARLE & CO (US) 1994-03-16 EP claimed
WO-1993023075-A1 TREATMENT OF VASCULAR LEAKAGE SYNDROME AND COLLAGENASE INDUCED DISEASE BY ADMINISTRATION OF MATRIX METALLOPROTEINASE INHIBITORS ONCOLOGIX, INC. (US) 1993-11-25 WO claimed
WO-1993021938-A1 METHODS FOR TREATING CANCER USING HIGH-DOSE EPIRUBICIN ADRIA LABORATORIES (US) 1993-11-11 WO claimed
US-5242901-A Bisdioxopiperazine compounds for cardiovascular disorders NEW YORK UNIVERSITY (US) 1993-09-07 US claimed
WO-1992008460-A1 BIS-DIOXOPIPERAZINES FOR TREATING LIVER TUMOURS WINDLESHAW ENTERPRISES LIMITED (GB) 1992-05-29 WO claimed
WO-1990012590-A1 TREATMENT OF OCULAR DISEASE BY MODULATION OF MATRIX METALLOPROTEINASES AND THEIR INHIBITOR STATE OF OREGON, STATE BOARD OF HIGHER EDUCATION, OREGON HEALTH SCIENCES UNIVERSITY (US) 1990-11-01 WO claimed
EP-0393575-A1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent G.D. Searle & Co. (US) 1990-10-24 EP claimed
US-4963679-A Process for preparing bis (3,5-dioxopiperazinyl) alkanes or alkenes ERBAMONT, INC. (US) 1990-10-16 US claimed
EP-0330381-A1 Process for preparing bis (3,5-dioxopiperazinyl) alkanes or alkenes ERBAMONT, INC. (US) 1989-08-30 EP claimed
US-4275063-A 1,2-BIS(3,5-DIOXOPIPERAZIN-YL)PROPANE FOR TREATMENT OF CANCER IN HUMANS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1981-06-23 US claimed