SCHEMBL9090100

SCHEMBL9090100

c1c[nH]c(-c2ccc3c(c2)CCN3)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.46
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
MTOR P42345 1/20 0.44
ADK P55263 1/20 0.44
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
S1PR1 P21453 2/20 0.40
S1PR3 Q99500 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP19A1 P11511 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
PIK3CD O00329 1/20 0.39
JAK2 O60674 1/20 0.38
JAK3 P52333 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29756191 0.78 DRD2 (0.63) DRD2DRD4KDM4EALDH1A1S1PR1
SCHEMBL28403784 0.78 DRD2 (0.63) DRD2DRD4KDM4EALDH1A1S1PR1
SCHEMBL27604500 0.77 NISCH (0.49) NISCHMTORADKKDM4EALDH1A1
SCHEMBL4525557 0.73 PDE3B (0.56) DRD2DRD4KDM4EALDH1A1PDE3B
SCHEMBL722191 0.72 NISCH (0.78) NISCHMTORADKKDM4EALDH1A1
SCHEMBL27586687 0.72 DYRK1A (0.50) NISCHMTORADKKDM4EALDH1A1
SCHEMBL26260184 0.71 NISCH (0.59) NISCHMTORADKKDM4EALDH1A1
SCHEMBL508525 0.71 TAAR1 (0.49) DRD2DRD4JAK2JAK3HRH3
SCHEMBL4533554 0.71 CDK2 (0.52) DRD2DRD4KDM4EALDH1A1S1PR1
SCHEMBL1436033 0.70 KDM4E (0.63) DRD2DRD4KDM4EALDH1A1PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5538973-A ANTIHISTAMINE, THROMBOXANE A2 ANTAGONIST KYOTO PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
EP-0597112-A1 NOVEL IMIDAZOLE DERIVATIVE, PHARMACEUTICAL USE THEREOF, AND INTERMEDIATE THEREFOR Kyoto Pharmaceutical Industries, Ltd. (JP) 1994-05-18 EP disclosed