SCHEMBL9095259

SCHEMBL9095259

COc1ccc(C)c2[nH]c(=O)c(C(C)C)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.46
PDE3A Q14432 2/20 0.46
ALDH1A1 P00352 6/20 0.43
KDM4E B2RXH2 4/20 0.43
HSD17B10 Q99714 4/20 0.43
TSHR P16473 1/20 0.43
NQO2 P16083 3/20 0.41
CYP19A1 P11511 2/20 0.41
HPGD P15428 3/20 0.40
TP53 P04637 1/20 0.40
PBK Q96KB5 1/20 0.39
TRPV1 Q8NER1 2/20 0.38
TNKS O95271 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
CNR2 P34972 2/20 0.37
GPR18 Q14330 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9095728 0.80 ALDH1A1 (0.39) ALDH1A1KDM4EHSD17B10HPGDCYP3A4
SCHEMBL9095099 0.79 HSD17B10 (0.33) PDE3BPDE3AALDH1A1KDM4EHSD17B10
SCHEMBL9095859 0.79 KDM4E (0.40) ALDH1A1KDM4EHSD17B10TSHRHPGD
SCHEMBL9095097 0.79 HSD17B10 (0.33) PDE3BPDE3AALDH1A1KDM4EHSD17B10
SCHEMBL9093518 0.79 DAO (0.43) ALDH1A1KDM4EHSD17B10TSHRHPGD
SCHEMBL9097057 0.79 PDE4B (0.38) ALDH1A1KDM4EHSD17B10HPGDCYP3A4
SCHEMBL24380300 0.78 KDM4E (0.41) PDE3BPDE3AALDH1A1KDM4EHSD17B10
SCHEMBL9096295 0.78 ALDH1A1 (0.54) PDE3BPDE3AALDH1A1KDM4EHSD17B10
SCHEMBL22408526 0.74 KDM4E (0.45) PDE3BPDE3AALDH1A1KDM4EHSD17B10
SCHEMBL22185212 0.73 CNR2 (0.48) ALDH1A1KDM4EHSD17B10NQO2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576324-A Quinoline derivatives or salt thereof and remedy for cardiac diseases containing the same KOWA CO., LTD. (JP) 1996-11-19 US disclosed
EP-0638571-A1 QUINOLINE DERIVATIVE OR SALT THEREOF AND REMEDY FOR CARDIAC DISEASES CONTAINING THE SAME KOWA CO. LTD. (JP) 1995-02-15 EP disclosed