SCHEMBL9099369

SCHEMBL9099369

O=[C]c1cccc2cc(C(=O)OCCc3ccccc3)ccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.52
ESR2 Q92731 1/20 0.52
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
L3MBTL1 Q9Y468 7/20 0.50
ATM Q13315 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
MMP12 P39900 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
GLA P06280 1/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9397888 0.80 ESR1 (0.65) ESR1ESR2NPC1RAB9AL3MBTL1
SCHEMBL7568065 0.78 L3MBTL1 (0.63) ESR1ESR2NPC1RAB9AL3MBTL1
SCHEMBL27327003 0.77 L3MBTL1 (0.69) ESR1ESR2NPC1RAB9AL3MBTL1
SCHEMBL4868189 0.76 LCK (0.54) ATMKDM4EMAPTHTTALDH1A1
SCHEMBL9670475 0.75 PTPN1 (0.62) KDM4EMAPTALDH1A1GLAHPGD
SCHEMBL4459400 0.75 ESR1 (0.86) ESR1ESR2NPC1RAB9AL3MBTL1
SCHEMBL9100113 0.74 ESR1 (0.69) ESR1ESR2NPC1RAB9AL3MBTL1
SCHEMBL10980613 0.74 ESR1 (0.69) ESR1ESR2NPC1RAB9AL3MBTL1
SCHEMBL9098921 0.74 TDP1 (0.54) NPC1RAB9ATDP1KDM4EMAPT
SCHEMBL7572516 0.74 L3MBTL1 (0.65) ESR1ESR2NPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0323441-B1 5-Fluorouracil derivatives OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
EP-0436902-B1 5-Fluorouracil derivatives OTSUKA PHARMA CO LTD (JP) 1995-06-28 EP disclosed
EP-0180897-B1 5-FLUOROURACIL DERIVATIVES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-08-07 EP disclosed
EP-0436902-A1 5-Fluorouracil derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-07-17 EP disclosed
US-4983609-A Anticancer agents OTSUKA PHARMACEUTICAL (JP) 1991-01-08 US disclosed
US-4864021-A ANTICARCINOGENIC AGENTS, ANTITUMOR AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-09-05 US disclosed
EP-0323441-A2 5-Fluorouracil derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-07-05 EP disclosed
EP-0180897-A2 5-Fluorouracil derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-05-14 EP disclosed